Corydalis Extract Tetrahydropalmatine (dl-THP)
Tetrahydropalmatine (THP), izwi kandi nka dl-THP, Corydalin hydrochloride, cyangwa Corydalin Tube Extract, ni ikintu gikomoka kuri isoquinoline alkaloid. Kivanwa mu kimera cy'igishinwa cyitwa Corydalis yanhusuo. THP ni ikintu kidafite ibara cyangwa umuhondo werurutse gifite uburyohe busharira gato kandi gishobora gushonga bwa dogere selisiyusi 147-149. Nta kintu na kimwe gishobora gushonga mu mazi ariko gishobora gushonga cyane muri ether, chloroform, na ethanol. Umunyu wayo wa hydrochloride na sulfate ushonga mu mazi.
THP yakozweho ubushakashatsi ku ngaruka zitandukanye z’imiti, harimo kugabanya ububabare, kugabanya ububabare, kurinda ubwonko, kurwanya guterana kw’imitsi, kurwanya ibisebe, kurwanya ikibyimba, no kurwanya ibiyobyabwenge. Bikekwa ko igira ingaruka nziza ku bubabare mu guhindura imikorere ya dopamine receptor kandi yagaragaje ubushobozi bwo kurinda uturemangingo kwangirika kw’imitsi. Byongeye kandi, THP yagaragaje ingaruka zo guterana kw’imitsi kandi yanakoreweho ubushakashatsi ku ngaruka zayo mu kuvura ibisebe, kubuza gukura kw’uturemangingo twa kanseri, no gufasha mu kuba imbata y’ibiyobyabwenge.
Muri rusange, Tetrahydropalmatine (dl-THP) ni ikinyabutabire gifite imiterere itandukanye y’imiti kandi cyakoreweho ubushakashatsi bwimbitse ku mikoreshereze yacyo ishobora gukoreshwa mu kuvura. Kubindi bisobanuro hamagaragrace@biowaycn.com.
Dore ibiranga Tetrahydropalmatine (THP) hamwe n'inyungu zayo ku buzima:
1. Imiterere y'uburibwe:THP igaragaza ingaruka zo kugabanya ububabare binyuze mu guhindura imikorere ya central dopamine receptor, igatanga ububabare butagira ubushobozi bugaragara bwo kubwibasira.
2. Ingaruka zo kurinda ubwonko:THP yagaragaje ubushobozi bwo kurinda uturemangingo kwangirika kw'imitsi, kugabanya apoptosis y'imitsi, no kugabanya urugero rwa glutamate mu bwonko, ibi bikaba bishobora kugira uruhare mu gutuma ubwonko burinda ubwonko.
3. Guteranya ibyuma birwanya uduce duto tw’amaraso:Byagaragaye ko THP ibuza platelets kwibumbira hamwe, ishobora kugabanya ibyago byo kubyimba kw'amaraso n'ibindi bibazo by'umutima n'imitsi.
4. Inkunga ku buzima bw'igifu:THP yagaragaje ingaruka zo kurwanya ibisebe kandi ishobora gufasha mu kugabanya isohoka rya aside mu gifu, igatanga ihumure ku bisebe byo mu gifu n'ibindi bifitanye isano na byo.
5. Iterambere rishobora kubaho mu kurwanya kanseri:THP yagaragaje ingaruka mbi ku turemangingo twa kanseri, bigaragaza ko ishobora kugira uruhare mu kubuza gukura kwa kanseri.
6. Imiterere yo kurwanya ibiyobyabwenge:THP yakozweho ubushakashatsi ku bushobozi bwayo bwo kugabanya ibimenyetso byo kureka ibiyobyabwenge bifitanye isano no kuba umuntu afite opioid n'ubusinzi, itanga icyizere cyo kuvura no gukumira kongera kubikoresha.
Ibi bintu bigaragaza inyungu zitandukanye ku buzima n'uburyo Tetrahydropalmatine (THP) ishobora gukoreshwa mu kuvura.
Tetrahydropydalin (dl-THP) iri mu bigize isoquinoline alkaloids kandi ni alkaloid, cyane cyane mu bwoko bwa Corydalis lucidum (Yan Hu Suo), ariko no mu bindi bimera nka Stephania rotunda. Ibi bimera bifite ikoreshwa gakondo mu buvuzi bw'ibimera bw'Abashinwa.Corydalis ni ikimera cy’ibimera kiramba, gifite uburebure bwa santimetero 10 kugeza kuri 20, gifite ibirayi by’uruziga. Inkingi zacyo zo hejuru y’ubutaka ni ngufi kandi zoroshye, zifite uburebure hejuru y’ishingiro. Amababi y’ibanze n’amababi ya cauline asa mu miterere, hamwe n’ibibabi; amababi ya cauline arasimburana, afite amababi 2 na 3 afatanye. Ibabi rya kabiri rikunze gucikamo ibice byose kandi rifite ibice birebire. Amababi mato ni uburebure burambuye, uburebure burambuye, cyangwa uburebure burambuye. Ifite umurongo, ifite uburebure bwa santimetero 2, ifite umutwe ugororotse cyangwa utyaye n’impande nziza. Ishurwe ryayo rifite ishusho nk’iya raceme, rifite amababi aheruka cyangwa ahanganye; uduce duto dufite imiterere ya lanceolate; indabyo ni umutuku-umutuku kandi zikura ku buryo butambitse ku duti duto, dufite uburebure bwa mm 6; agace ka kari kagwa kare; indabyo ni 4 naho utundi duce two hanze ni 2. Ibice ni binini gato, bifite impande z’umutuku n’ubururu-umutuku hagati. Hari igice kimwe cyo hejuru, kandi umurizo urambuka ukagera ku gice kirekire. Uburebure bwa spur bugira hafi kimwe cya kabiri cy’uburebure bwose. Ibice bibiri by'imbere ni bito ugereranyije n'ibice bibiri byo hanze. Igice cyo hejuru ni ibara ry'umukara n'umuhengeri kandi cyakize, naho igice cyo hasi ni umutuku; Inkingi ni 6, kandi uduce dufatanye mu duce tubiri, buri kimwe gifite anthers 3; intanga ngabo ni ngufi kandi nto, kandi stigma ni 2, nk'ikinyugunyugu gito. Imbuto zayo ni agace gato. Corydalis ikorerwa cyane cyane mu misozi cyangwa mu byatsi. Uduce twinshi tuyibyaza umusaruro turimo Zhejiang, Hebei, Shandong, Jiangsu, n'ahandi.
| Isesengura | Ibisobanuro |
| Isuzuma | Tetrahydropalmatine ≥98% |
| Isura | Ifu y'umuhondo woroshye kuva ku mweru |
| Ivu | ≤0.5% |
| Ubushuhe | ≤5.0% |
| Imiti yica udukoko | Ububi |
| Ibyuma biremereye | ≤10ppm |
| Pb | ≤2.0ppm |
| As | ≤2.0ppm |
| Impumuro mbi | Ibiranga |
| Ingano y'uduce duto | 100% kugeza kuri 80 mesh |
| Ibinyabuzima: | |
| Igiteranyo cya bagiteri | ≤1000cfu/g |
| Ibihumyo | ≤100cfu/g |
| Salmgosella | Ububi |
| Coli | Ububi |
Dore inganda zikoresha ibikoresho bya Tetrahydropalmatine (THP):
1. Imiti:THP ikoreshwa mu nganda zikora imiti mu guteza imbere imiti yo kugabanya ububabare n'imiti irinda ubwonko.
2. Ibinyabutabire:THP ikoreshwa mu nganda z'intungamubiri mu gukora inyunganiramirire zigamije kugabanya ububabare no gufasha ubuzima bw'igifu.
3. Ikoranabuhanga mu by'ibinyabuzima:THP isanga ikoreshwa muri biotechnology mu bushakashatsi ku miti igabanya udukoko two mu maraso ndetse n'ibindi bishobora kuba imiti ishobora kuvura kanseri.
4. Ubuvuzi:THP ishyirwa mu bicuruzwa by’ubuvuzi mu kuvura indwara zo kubagwa n’ibimenyetso byo kubireka bifitanye isano no gukoresha opioid n’ibitera imbaraga.
5. Ibikoresho byo mu rwego rwo hejuru:THP irasuzumwa mu bijyanye n'ubwiza bw'uruhu kugira ngo hamenyekane niba uruhu rushobora kumererwa neza ndetse n'uburyo bwo kugabanya ububyimbirwe.
Izi nganda zigaragaza uburyo butandukanye bwo gukoresha Tetrahydropalmatine (THP) mu iterambere ry’ibicuruzwa bitandukanye no mu bushakashatsi.
Ibicuruzwa byacu bikorwa hakoreshejwe ingamba zikomeye zo kugenzura ubuziranenge kandi bikurikiza amahame yo hejuru y’uburyo bwo gukora. Dushyira imbere umutekano n’ubwiza bw’ibicuruzwa byacu, tukareba ko byujuje ibisabwa n’amategeko n’ibyemezo by’inganda. Uku kwiyemeza ubuziranenge kugamije gushyiraho icyizere n’icyizere mu kwizerwa kw’ibicuruzwa byacu. Uburyo rusange bwo gukora ni ubu bukurikira:
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